
Name: | Darifenacin N-Oxide |
Catalogue No. | VL1530009 |
CAS No. | 1391080-40-2 |
Molecular Formula | C₂₈H₃₀N₂O₃ |
Molecular Weight | 442.55 |
Status | In-stock |
IUPAC Name | (3S)-3-(2-amino-2-oxo-1,1-diphenylethyl)-1-(2-(2,3-dihydrobenzofuran-5-yl)ethyl)pyrrolidine 1-oxide |
Description | Darifenacin N-Oxide (CAS No.: 1391080-40-2) or (3S)-3-(2-amino-2-oxo-1,1-diphenylethyl)-1-(2-(2,3-dihydrobenzofuran-5-yl)ethyl)pyrrolidine 1-oxide is an N-Oxide metabolite of Darifenacin which is a pure antimuscarinics compound. Although the clinical efficacy has been proven to be high its use is limited by various adverse effects. |
References | Scheepe, J. R., et al. “Effects of Propiverine and Its Metabolite Propiverine-N-Oxide on Bladder Contraction and Salivation in Mini Pigs.” Urologia Internationalis, vol. 81, no. 4, 2008, pp. 468–73,https://doi.org/10.1159/000167849. |